

{"id":15489,"date":"2013-12-11T11:33:49","date_gmt":"2013-12-11T03:33:49","guid":{"rendered":"https:\/\/case.ntu.edu.tw\/blog\/?p=15489"},"modified":"2017-07-27T10:47:37","modified_gmt":"2017-07-27T02:47:37","slug":"%e6%94%b9%e8%ae%8a%e8%85%a6%e5%85%a7%e5%8f%97%e9%ab%94%e6%b4%bb%e6%80%a7%ef%bc%8c%e6%9c%89%e6%95%88%e5%90%91%e6%af%92%e7%99%ae%e8%aa%aabye-bye%ef%bc%81","status":"publish","type":"post","link":"https:\/\/case.ntu.edu.tw\/blog\/?p=15489","title":{"rendered":"\u3010\u91ab\u5b78\u65b0\u77e5\u3011\u6539\u8b8a\u8166\u5167\u53d7\u9ad4\u6d3b\u6027\uff0c\u6709\u6548\u5411\u6bd2\u766e\u8aaaBYE BYE\uff01"},"content":{"rendered":"<p><strong>\u7de8\u8b6f\uff5c<\/strong>\u67ef\u5b97\u4f51<\/p>\n<p><span style=\"color: #333399;\"><b><strong>\u25a0<\/strong>\u7814\u7a76<\/b><b>\u767c\u73fe\uff0c\u63d0\u5347\u5c0f\u9f20\u8166\u5167\u9ea9\u80fa\u9178\u53d7\u9ad4\uff08<\/b><b>glutamate receptor<\/b><b>\uff09\u7684\u6d3b\u6027\uff0c\u80fd\u8b93\u5c0f\u9f20\u5728\u6212\u4e86\u53e4\u67ef\u9e7c\u4e4b\u5f8c\uff0c\u5fc3\u88e1\u4e0d\u6703\u7e7c\u7e8c\u60f3\u6bd2\u54c1\u60f3\u500b\u6c92\u5b8c\u3002<\/b><\/span><b><i><\/i><\/b><\/p>\n<p><a href=\"http:\/\/case.ntu.edu.tw\/blog\/wp-content\/uploads\/2013\/12\/rat.jpg\"><img fetchpriority=\"high\" decoding=\"async\" class=\"alignleft size-full wp-image-15490\" src=\"http:\/\/case.ntu.edu.tw\/blog\/wp-content\/uploads\/2013\/12\/rat.jpg\" alt=\"rat\" width=\"310\" height=\"174\" srcset=\"https:\/\/case.ntu.edu.tw\/blog\/wp-content\/uploads\/2013\/12\/rat.jpg 310w, https:\/\/case.ntu.edu.tw\/blog\/wp-content\/uploads\/2013\/12\/rat-300x168.jpg 300w\" sizes=\"(max-width: 310px) 100vw, 310px\" \/><\/a><\/p>\n<p>\u53e4\u67ef\u9e7c\u6210\u766e\u60a3\u8005\u6703\u4ee4\u91ab\u8b77\u4eba\u54e1\u611f\u5230\u68d8\u624b\uff0c\u6b63\u662f\u56e0\u70ba\u9019\u4e9b\u4eba\u53ea\u8981\u63a5\u6536\u5230\u8207\u300c\u6bd2\u54c1\u300d\u6709\u95dc\u7684\u8a0a\u606f\uff0c\u766e\u982d\u5c31\u5f88\u53ef\u80fd\u5fa9\u767c\uff0c\u800c\u5c0f\u9f20\u548c\u4eba\u985e\u4e00\u6a23\uff0c\u4e5f\u6709\u985e\u4f3c\u7684\u53e4\u67ef\u9e7c\u6212\u65b7\u75c7\u72c0\u3002\u4e0d\u904e\uff0c\u4f0a\u5229\u8afe\u5dde\u5317\u829d\u52a0\u54e5\u5e02\uff08North Chicago\uff09\u7f85\u838e\u7433\uff0e\u5bcc\u862d\u514b\u6797\u91ab\u5b78\u8207\u79d1\u5b78\u5927\u5b78\uff08Rosalind Franklin University of Medicine and Science\uff09\u7684\u7814\u7a76\u4eba\u54e1\u6700\u8fd1\u767c\u73fe\uff0c\u4e00\u65e6\u589e\u5f37\u5c0f\u9f20\u5927\u8166\u5167\u67d0\u500b\u9ea9\u80fa\u9178\u53d7\u9ad4\u7684\u6d3b\u6027\uff0c\u5c31\u80fd\u6291\u5236\u5176\u6212\u65b7\u75c7\u72c0\u3002\u9019\u9805\u7531\u746a\u8389\u5b89\uff0e\u6c83\u723e\u592b\uff08Marina Wolf\uff09\u3001Kuei Tseng\u7b49\u4eba\u9032\u884c\u7684\u7814\u7a76\uff0c\u5df2\u7d93\u5728\u300a\u81ea\u7136\u795e\u7d93\u79d1\u5b78\u300b\uff08<i>Nature Neuroscience<\/i>\uff09\u671f\u520a\u4e2d\u767c\u8868\u4e86\u3002<\/p>\n<p><b>\u766e\u982d\u958b\u95dc<\/b><\/p>\n<p>\u6c83\u723e\u592b\u548cTseng\u7387\u9818\u7684\u7814\u7a76\u5718\u968a\u767c\u73fe\uff0c\u5c0f\u9f20\u63a5\u6536\u53e4\u67ef\u9e7c\u76f8\u95dc\u8a0a\u606f\u5f8c\u4e4b\u6240\u4ee5\u840c\u751f\u766e\u982d\uff0c\u5176\u5be6\u8207\u5927\u8166\u4f0f\u9694\u6838\uff08nucleus accumbens, NAcc\uff09\u4e2d\u67d0\u4e00\u7f55\u898b\u7684\u9ea9\u80fa\u9178\u53d7\u9ad4\uff0c\u4e5f\u5c31\u662f\u9223\u96e2\u5b50\u901a\u900f\u578bAMPA\u53d7\u9ad4\uff08Ca<sup>2+<\/sup>-permeable AMPA receptor\uff0c\u4ee5\u4e0b\u7c21\u7a31CP-AMPAR\uff09\u5927\u91cf\u589e\u52a0\u6709\u95dc\u3002\u540c\u6642\u4ed6\u5011\u4e5f\u767c\u73fe\uff0c\u53ea\u8981\u63d0\u5347\u53e6\u4e00\u7a2e\u9ea9\u80fa\u9178\u53d7\u9ad4\u2014\u2014\u4ee3\u8b1d\u578b\u9ea9\u80fa\u9178\u53d7\u9ad41\uff08metabotropic glutamate receptor 1, \u4ee5\u4e0b\u7c21\u7a31mGluR1\uff09\u7684\u6d3b\u6027\uff0c\u5c31\u80fd\u5c07CP-AMPAR\u81ea\u4f0f\u9694\u6838\u4e2d\u7684\u795e\u7d93\u7a81\u89f8\uff08synapse\uff09\u6e05\u9664\u3002\u4e8b\u5be6\u4e0a\uff0c\u7121\u8ad6\u4f4d\u65bc\u5927\u8166\u54ea\u4e00\u5340\uff0cCP-AMPAR\u7684\u4f5c\u7528\u90fd\u76f8\u7576\u4e00\u81f4\uff0c\u800c\u5be6\u9a57\u8b49\u660e\uff0c\u53ea\u8981\u589e\u5f37mGluR1\u7684\u6d3b\u6027\uff0c\u5c31\u80fd\u58d3\u5236CP-AMPAR\u7684\u4f5c\u7528\uff0c\u9054\u5230\u53bb\u9664\u766e\u982d\u7684\u6548\u679c\u4e86\u3002<\/p>\n<p>\u672a\u53c3\u8207\u7814\u7a76\u8a08\u756b\u7684\u745e\u58eb\u65e5\u5167\u74e6\u5927\u5b78\uff08University of Geneva\uff09\u795e\u7d93\u79d1\u5b78\u8207\u795e\u7d93\u91ab\u5b78\u6559\u6388\u514b\u91cc\u65af\u63d0\u5b89\uff0e\u5442\u820d\u723e\uff08Christian L\u00fcscher\uff09\u8868\u793a\uff0c\u9019\u9805\u6700\u65b0\u7814\u7a76\uff1a\u300c\u5167\u5bb9\u975e\u5e38\u5b8c\u5584\uff0c\u5c07mGluR\u5c0d\u6210\u766e\u7684\u63a7\u5236\u6548\u679c\u7814\u7a76\u5f97\u6e05\u6e05\u695a\u695a\u3002\u300d\u5442\u820d\u723e\u6559\u6388\u9084\u8868\u793a\uff0cCP-AMPAR\u7684\u5b58\u5728\u6642\u9593\u76f8\u7576\u77ed\uff0c\u4f46\u6b64\u6642\u5927\u8166\u7684\u53ef\u5851\u6027\u4e5f\u8b8a\u5f97\u76f8\u7576\u9ad8\uff1a\u300c\u6216\u8a31\u9019\u5c31\u662f\u6bd2\u54c1\u50b7\u8166\u7684\u6642\u6a5f\u3002\u300d<!--more--><\/p>\n<p><b>\u4e00\u89e3\u5c0f\u9f20\u766e\u982d<\/b><\/p>\n<p>\u9019\u9805\u7814\u7a76\u4ee5\u5c0f\u9f20\u70ba\u5be6\u9a57\u5c0d\u8c61\uff0c\u9996\u5148\u5c07\u751f\u7406\u98df\u9e7d\u6c34\u53ca\u53e4\u67ef\u9e7c\u900f\u904e\u5c0e\u7ba1\u6ce8\u5165\u4e0d\u540c\u7684\u76d2\u5b50\u88e1\uff0c\u518d\u6293\u8d77\u5c0f\u9f20\uff0c\u5c07\u5176\u9f3b\u5b50\u6e4a\u5165\u4e0d\u540c\u7684\u76d2\u5b50\u88e1\uff0c\u6b64\u6642\u4e5f\u6703\u555f\u52d5\u76d2\u4e2d\u7684\u71c8\u5149\u3002\u6bcf\u5929\u9032\u884c\u524d\u8ff0\u6b65\u9a5f\u516d\u5c0f\u6642\uff0c\u7d93\u904e\u5341\u5929\u9069\u61c9\u671f\u5f8c\uff0c\u4fbf\u9032\u5165\u6212\u65b7\u6642\u671f\uff0c\u8207\u60a3\u6bd2\u766e\u7684\u4eba\u985e\u66ab\u6642\u4e0d\u78b0\u6bd2\u7684\u505a\u6cd5\u53ef\u8aaa\u662f\u4e00\u6a21\u4e00\u6a23\u3002\u9019\u6642\uff0c\u76d2\u4e2d\u5df2\u7d93\u6c92\u6709\u53e4\u67ef\u9e7c\u4e86\uff0c\u7814\u7a76\u4eba\u54e1\u958b\u59cb\u89c0\u5bdf\u5c0f\u9f20\u5982\u4f55\u5c0d\u6bd2\u54c1\u76f8\u95dc\u8a0a\u865f\uff0c\u4e5f\u5c31\u662f\u9f3b\u5b50\u5165\u76d2\u6642\u9ede\u4eae\u7684\u71c8\u5149\u7522\u751f\u53cd\u61c9\u3002\u4ed6\u5011\u767c\u73fe\uff0c\u60a3\u6709\u6bd2\u766e\u7684\u5c0f\u9f20\u4e00\u5982\u9810\u671f\uff0c\u6703\u56e0\u63a5\u53d7\u76f8\u95dc\u8a0a\u865f\u840c\u751f\u766e\u982d\u3002\u800c\u7576\u7814\u7a76\u4eba\u54e1\u7d66\u5c0f\u9f20\u65bd\u6253\u67d0\u7a2emGluR1\u6b63\u5411\u7570\u4f4d\u8abf\u63a7\u5206\u5b50\uff08positive allosteric modulator\uff09\uff0c\u4e5f\u5c31\u662f\u540d\u70baSYN119\u7684\u85e5\u7269\u6642\uff0c\u7121\u8ad6\u662f\u671d\u8179\u819c\u5167\u6ce8\u5c04\uff0c\u6216\u76f4\u63a5\u671d\u4f0f\u9694\u6838\u6ce8\u5c04\uff0c\u5c0f\u9f20\u5728\u6212\u65b7\u5f8c\u7b2c45\u5929\u7684\u6210\u766e\u73fe\u8c61\u5c31\u6703\u6e1b\u5c11\u8a31\u591a\uff0c\u6bd4\u4e0d\u662f\u65bd\u6253SYN119\u7684\u63a7\u5236\u7d44\u5c0f\u9f20\u4f86\u5f97\u660e\u986f\u3002\u986f\u7136\uff0c\u53ea\u8981\u589e\u5f37mGluR1\u7684\u6d3b\u6027\uff0c\u5c31\u80fd\u964d\u4f4e\u5c0f\u9f20\u63a5\u6536\u53e4\u67ef\u9e7c\u76f8\u95dc\u8a0a\u865f\u6642\u840c\u751f\u7684\u766e\u982d\u3002<\/p>\n<p>\u5be6\u9a57\u904e\u5f8c\uff0c\u7814\u7a76\u4eba\u54e1\u5c07\u5be6\u9a57\u7d44\u53ca\u63a7\u5236\u7d44\u5c0f\u9f20\u7684\u5927\u8166\u5207\u7247\uff0c\u4e26\u900f\u904e\u96fb\u751f\u7406\u5b78\uff08electrophysiology\uff09\u65b9\u5f0f\u89c0\u5bdf\u5207\u7247\uff0c\u4ee5\u8b49\u660e\u6ce8\u5c04SYN119\u4e4b\u5f8c\uff0c\u5c0f\u9f20\u8166\u4f0f\u9694\u6838\u5167\u7684CP-AMPAR\u6d3b\u6027\u78ba\u5be6\u964d\u4f4e\uff0c\u800c\u4e14\u6548\u671f\u53ef\u905424\u5c0f\u6642\u3002\u6b64\u5916\uff0c\u7814\u7a76\u4eba\u54e1\u9084\u53cd\u5411\u64cd\u4f5c\uff0c\u5148\u5728\u6212\u65b7\u524d\u671f\u4ee5\u62ee\u6297\u5291\u6e1b\u5c11\u4f0f\u9694\u6838\u5167\u7684mGluR1\uff0c\u518d\u89c0\u5bdf\u6212\u65b7\u671f\u9593\uff0cCP-AMPAR\u6578\u91cf\u662f\u5426\u6703\u589e\u52a0\uff0c\u7d50\u679c\u986f\u793a\uff0cCP-AMPAR\u7684\u78ba\u99ac\u4e0a\u589e\u52a0\uff0c\u7531\u6b64\u53ef\u8b49\uff0cmGluR1\u80fd\u6709\u6548\u6291\u5236CP-AMPAR\uff0c\u9054\u5230\u58d3\u6291\u766e\u982d\u7684\u6548\u679c\u3002<\/p>\n<p>\u6c83\u723e\u592b\u8868\u793a\uff1a\u300c\u9019\u4e9b\u6212\u65b7\u75c7\u72c0\uff0c\u90fd\u662f\u56e0\u70ba\u795e\u7d93\u5143\u88e1\u7684\u67d0\u4e9b\u90e8\u5206\u5728\u4f5c\u602a\uff0c\u4e0d\u53ea\u548cCP-AMPAR\u6709\u95dc\uff0c\u4e5f\u6d89\u53ca\u5176\u4ed6\u7684\u7a81\u89f8\u529f\u80fd\u3002mGluR1\u662f\u6709\u6291\u5236\u766e\u982d\u7684\u6548\u679c\uff0c\u4f46\u6211\u500b\u4eba\u89ba\u5f97\uff0c\u5f8c\u9762\u9084\u6709\u66f4\u591a\u8907\u96dc\u7684\u6a5f\u5236\u5728\u4f5c\u7528\u3002\u300d<\/p>\n<p><b>\u773e\u671b\u6240\u6b78\u7684\u5206\u5b50<\/b><\/p>\n<p>\u540c\u6a23\u672a\u53c3\u8207\u7814\u7a76\u8a08\u756b\u7684\u611b\u8377\u83ef\u5927\u5b78\uff08University of Iowa\uff09\u5fc3\u7406\u5b78\u52a9\u7406\u6559\u6388\u96f7\u6069\uff0e\u62c9\u9b6f\u7c73\u723e\uff08Ryan LaLumiere\uff09\u5247\u8868\u793a\uff1a\u300c\u9019\u9805\u7814\u7a76\u7684\u7368\u5230\u4e4b\u8655\uff0c\u5728\u65bc\u5176\u7d50\u679c\u53ef\u80fd\u5c0d\u81e8\u5e8a\u6cbb\u7642\u53ca\u8f49\u8b6f\u91ab\u5b78\u5927\u6709\u52a9\u76ca\u3002\u4e00\u822c\u800c\u8a00\uff0c\u6211\u5011\u5f88\u96e3\u91dd\u5c0d\u4eba\u8166\u4e2d\u7684\u67d0\u500b\u53d7\u9ad4\u4e0b\u624b\uff0c\u56e0\u70ba\u4e00\u65e6\u9032\u884c\u8655\u7f6e\uff0c\u5f88\u6709\u53ef\u80fd\u5e72\u64fe\u5176\u4ed6\u8166\u5340\u7684\u529f\u80fd\uff0c\u4f46\u9019\u7a2e\u8abf\u63a7\u5206\u5b50\u6709\u5176\u91dd\u5c0d\u6027\uff0c\u526f\u4f5c\u7528\u4e0d\u592a\u591a\u3002\u300d<\/p>\n<p>\u5c0d\u65bc\u7570\u4f4d\u8abf\u63a7\u5206\u5b50\u7684\u529f\u80fd\uff0c\u9054\u62c9\u65af\u5e02\u5fb7\u5dde\u5927\u5b78\u897f\u5357\u91ab\u5b78\u4e2d\u5fc3\uff08University of Texas Southwestern Medical Center\uff09\u7cbe\u795e\u91ab\u5b78\u6559\u6388\u5927\u885b\uff0e\u745f\u592b\uff08David 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\/>\n--<\/p>\n<pre><span style=\"color: #333333;\"> \u7814\u7a76\u51fa\u8655\uff1a<strong><a href=\"http:\/\/www.the-scientist.com\/?articles.view\/articleNo\/38431\/title\/Suppressing-Drug-Seeking-Behaviors\/\">Suppressing Drug-Seeking Behaviors<\/a><\/strong><\/span><\/pre>\n<p><span style=\"color: #333399;\"><strong><strong>\u8cac\u4efb\u7de8\u8f2f\uff1aKerina Huang<\/strong><\/strong><\/span><\/p>\n","protected":false},"excerpt":{"rendered":"<p>\u7de8\u8b6f\uff5c\u67ef\u5b97\u4f51 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